gpss_a_1653870_sm1681.docx (4.52 MB)
Facile synthesis of novel Mono- and Bis-N-sulfamoylamidines
journal contribution
posted on 2019-08-16, 12:15 authored by Ye Xuan-Wu, Abudureheman WusimanMono- and bis-N-sulfamoylamidines have been efficiently synthesized by the direct condensation of sulfamides and amides in the presence of phosphorus oxychloride via electrophilic activation. The scope of this reaction is discussed, and detailed synthetic studies show that the desired products are generated in high yields under mild conditions.